~65 spots leftby Jun 2027

Naltrexone/Bupropion for Obesity

Recruiting in Palo Alto (17 mi)
JK
Overseen byJudith Korner, MD,PhD
Age: 18+
Sex: Any
Travel: May Be Covered
Time Reimbursement: Varies
Trial Phase: Phase 4
Recruiting
Sponsor: Columbia University
Must be taking: Naltrexone/bupropion
Must not be taking: Dopamine agonists, Opioid analgesics
Disqualifiers: Diabetes, Cardiovascular disease, Seizures, others
No Placebo Group
Prior Safety Data
Approved in 3 Jurisdictions

Trial Summary

What is the purpose of this trial?

The goal of this clinical trial is to understand if genetic variations are associated with the amount of weight loss with diet and while taking an FDA-approved medication for weight loss. The main question\[s\] it aims to answer are: * In Aim One, the investigators propose to rigorously test the hypothesis that presence of the Taq1A A1+ polymorphism is associated with greater weight loss with NB compared with the A1- genotype. * In Aim Two, the investigators will explore other genetic polymorphisms that might influence the efficacy of NB such as the fat mass and obesity-associated (FTO) gene which modulates DRD2 signaling, as carriers of risk alleles in both the FTO and ANKK1 gene demonstrate altered responses to reward-learning tasks associated with negative outcomes. Participants will be in the study for 40 weeks, which consists of two phases: 1. From baseline to week 12, participants will receive individual nutritional counseling on a calorie restricted diet. This phase includes in-person visits, blood tests, an EKG, vital signs, questionnaires, body weight, and nutritional visits. 2. From week 12 to week 40, participants will continue to receive dietary counseling and will receive treatment with naltrexone/bupropion for 28 weeks. This phase includes in-person and phone visits, blood tests, vital signs, questionnaires, body weight, and nutritional visits.

Will I have to stop taking my current medications?

Yes, you may need to stop taking certain medications. The trial excludes participants using dopamine agonists, opioid analgesics, antipsychotics, antidepressants, neuroleptics, naltrexone, diabetes medications, and MAO inhibitors within 14 days prior to screening. It also excludes those using weight loss medication within the prior six months.

What evidence supports the effectiveness of the drug naltrexone/bupropion for obesity?

Research shows that naltrexone/bupropion can lead to significant weight loss and improved quality of life in patients with genetic obesity, as seen in a case where a patient lost 48.9 kg over 17 months. Additionally, a study found that individuals with a specific genetic variant experienced greater weight loss with this drug, suggesting it may be more effective for certain people.12345

Is Naltrexone/Bupropion safe for humans?

Research shows that Naltrexone/Bupropion does not increase the risk of major heart-related events in humans, suggesting it is generally safe for use.12367

How does the drug naltrexone/bupropion work for obesity?

Naltrexone/bupropion is unique because it combines two drugs that work on the brain to help control appetite and cravings, which can lead to significant weight loss. This combination is particularly effective for people with certain genetic traits, like the Taq1A variant, and has shown success where other treatments have failed.12389

Research Team

JK

Judith Korner, MD,PhD

Principal Investigator

Columbia University

Eligibility Criteria

This trial is for men and women aged 18-65 with obesity, defined as a BMI of 30-50, or overweight individuals (BMI 27-29.99) with certain weight-related health issues like controlled high blood pressure, cholesterol problems, sleep apnea, or joint arthritis.

Inclusion Criteria

My BMI is between 30-50, or 27-29.99 with a weight-related health issue.
I am between 18 and 65 years old.

Exclusion Criteria

My current weight is more than 5% less than my highest weight ever.
I am not taking drugs that interfere with CYP2B6.
An affirmative answer to any question in the Columbia-Suicide Severity Rating Scale
See 17 more

Trial Timeline

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Nutritional Counseling

Participants receive individual nutritional counseling on a calorie restricted diet, including in-person visits, blood tests, an EKG, vital signs, questionnaires, body weight, and nutritional visits

12 weeks
In-person visits

Treatment with Naltrexone/Bupropion

Participants continue dietary counseling and receive treatment with naltrexone/bupropion, including in-person and phone visits, blood tests, vital signs, questionnaires, body weight, and nutritional visits

28 weeks
In-person and phone visits

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

Treatment Details

Interventions

  • Genetics and Response to Naltrexone/Bupropion (Other)
Trial OverviewThe study tests if genetic differences affect how well people lose weight on a calorie-restricted diet and the FDA-approved medication Naltrexone-Bupropion (NB). It's divided into three phases over one year: initial diet counseling and assessments; continued dieting plus NB treatment; then a wash-out period to see if genetics relate to maintaining weight loss.
Participant Groups
1Treatment groups
Experimental Treatment
Group I: All participantsExperimental Treatment1 Intervention
Calorie restricted diet and treatment with Naltrexone/Bupropion

Find a Clinic Near You

Research Locations NearbySelect from list below to view details:
Columbia University Medical CenterNew York, NY
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Who Is Running the Clinical Trial?

Columbia University

Lead Sponsor

Trials
1529
Patients Recruited
2,832,000+

National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK)

Collaborator

Trials
2513
Patients Recruited
4,366,000+

Findings from Research

Successful naltrexone-bupropion treatment after several treatment failures in a patient with severe monogenic obesity.Welling, MS., Mohseni, M., van der Valk, ES., et al.[2023]
A randomized, phase 3 trial of naltrexone SR/bupropion SR on weight and obesity-related risk factors (COR-II).Apovian, CM., Aronne, L., Rubino, D., et al.[2021]
Weight-loss response to naltrexone/bupropion is modulated by the Taq1A genetic variant near DRD2 (rs1800497): A pilot study.Mullally, JA., Chung, WK., LeDuc, CA., et al.[2022]
Pharmacogenetics of obesity drug therapy.Guzman, AK., Ding, M., Xie, Y., et al.[2021]
Addictive genes and the relationship to obesity and inflammation.Heber, D., Carpenter, CL.[2021]
Use of Contrave, Naltrexone with Bupropion, Bupropion, or Naltrexone and Major Adverse Cardiovascular Events: A Systematic Literature Review.Dahlberg, S., Chang, ET., Weiss, SR., et al.[2022]
Naltrexone/Bupropion ER (Contrave): Newly Approved Treatment Option for Chronic Weight Management in Obese Adults.Sherman, MM., Ungureanu, S., Rey, JA.[2020]
In a 56-week study involving 505 overweight or obese individuals with type 2 diabetes, the combination of naltrexone and bupropion (NB) led to significantly greater weight loss (-5.0% vs. -1.8%) and a higher percentage of participants achieving at least 5% weight loss compared to placebo (44.5% vs. 18.9%).
NB therapy also improved glycemic control, with a greater reduction in HbA1c levels (-0.6% vs. -0.1%) and a higher proportion of patients reaching HbA1c <7% (44.1% vs. 26.3%), although it was associated with increased gastrointestinal side effects like nausea and vomiting.
Effects of naltrexone sustained-release/bupropion sustained-release combination therapy on body weight and glycemic parameters in overweight and obese patients with type 2 diabetes.Hollander, P., Gupta, AK., Plodkowski, R., et al.[2022]
Bupropion and naltrexone: a review of their use individually and in combination for the treatment of obesity.Plodkowski, RA., Nguyen, Q., Sundaram, U., et al.[2019]

References

Successful naltrexone-bupropion treatment after several treatment failures in a patient with severe monogenic obesity. [2023]
A randomized, phase 3 trial of naltrexone SR/bupropion SR on weight and obesity-related risk factors (COR-II). [2021]
Weight-loss response to naltrexone/bupropion is modulated by the Taq1A genetic variant near DRD2 (rs1800497): A pilot study. [2022]
Pharmacogenetics of obesity drug therapy. [2021]
Addictive genes and the relationship to obesity and inflammation. [2021]
Use of Contrave, Naltrexone with Bupropion, Bupropion, or Naltrexone and Major Adverse Cardiovascular Events: A Systematic Literature Review. [2022]
Naltrexone/Bupropion ER (Contrave): Newly Approved Treatment Option for Chronic Weight Management in Obese Adults. [2020]
Effects of naltrexone sustained-release/bupropion sustained-release combination therapy on body weight and glycemic parameters in overweight and obese patients with type 2 diabetes. [2022]
Bupropion and naltrexone: a review of their use individually and in combination for the treatment of obesity. [2019]