~11 spots leftby Apr 2027

Darolutamide for Salivary Gland Cancer

Recruiting in Palo Alto (17 mi)
+29 other locations
Alan L. Ho, MD, PhD - MSK Head and Neck ...
Overseen byAlan L Ho, MD, PhD
Age: 18+
Sex: Any
Travel: May Be Covered
Time Reimbursement: Varies
Trial Phase: Phase 2
Recruiting
Sponsor: National Cancer Institute (NCI)
Must be taking: Androgen inhibitors, GnRH agonists
Must not be taking: P-gp inducers, CYP3A inducers
Disqualifiers: Vascular events, Allergic reactions, others
No Placebo Group
Prior Safety Data

Trial Summary

What is the purpose of this trial?

This phase II trial tests how well darolutamide and leuprolide acetate work in treating patients with androgen receptor positive salivary cancer that has spread from where it first started (primary site) to other places in the body (metastatic), cannot be removed by surgery (unresectable) or that has come back after a period of responding to prior therapy (recurrent). Darolutamide is in a class of medications called androgen receptor inhibitors. It works by blocking the effects of androgen (a male reproductive hormone) to stop the growth and spread of cancer cells. Leuprolide acetate is in a class of medications called gonadotropin-releasing hormone (GnRH) agonists. It works by decreasing the amount of certain hormones in the body. Giving darolutamide in combination with leuprolide acetate may help to stop the growth of tumor cells that need androgens to grow or shrink them.

Do I need to stop my current medications to join the trial?

The trial does not specify if you need to stop taking your current medications, but it does exclude patients on certain medications that interact with the trial drugs. It's important to discuss your current medications with the trial team to ensure there are no interactions.

What data supports the effectiveness of the drug Darolutamide for treating salivary gland cancer?

Darolutamide has been shown to be effective in treating prostate cancer by blocking androgen receptors, which are proteins that can promote cancer growth. While there is no direct evidence for its use in salivary gland cancer, its success in prostate cancer suggests it might help in other cancers that rely on similar growth pathways.12345

Is darolutamide safe for humans?

Darolutamide has been shown to be generally safe in humans, with a manageable tolerability profile in clinical trials for prostate cancer. It is well tolerated and has a low risk of causing central nervous system-related side effects, such as seizures, which are common with similar drugs.13567

How is the drug Darolutamide unique for treating salivary gland cancer?

Darolutamide is unique because it is a second-generation androgen receptor inhibitor that does not cross the blood-brain barrier, reducing the risk of seizures, and it can inhibit resistant cancer cell variants. While primarily used for prostate cancer, its novel mechanism may offer new hope for salivary gland cancer, which lacks standard treatments.13589

Research Team

Alan L. Ho, MD, PhD - MSK Head and Neck ...

Alan L Ho, MD, PhD

Principal Investigator

JHU Sidney Kimmel Comprehensive Cancer Center LAO

Eligibility Criteria

Adults with advanced salivary gland cancer that has spread, can't be surgically removed, or has returned after treatment. Participants must have tumors responsive to androgen (a male hormone), measurable disease, acceptable organ function, no prior androgen-targeted therapy (except under certain conditions), and an ECOG performance status of <=2. They should not have severe heart issues or other illnesses that could affect the trial's safety.

Inclusion Criteria

I have had treatment for brain metastases.
Total bilirubin =< 1.5 x institutional upper limit of normal (ULN) (exception: patients with elevated bilirubin due to Gilbert's disease would be eligible for the trial)
My tumor can be safely biopsied.
See 17 more

Exclusion Criteria

Patients with uncontrolled intercurrent illness
Patients who are receiving any other investigational agents
I have had a stroke or heart attack in the last 6 months.
See 5 more

Trial Timeline

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive darolutamide orally twice daily and leuprolide acetate intramuscularly every 4 or 12 weeks. Cycles repeat every 28 days in the absence of disease progression or unacceptable toxicity.

Up to 1 year
Monthly visits for treatment and monitoring

Follow-up

Participants are monitored for safety and effectiveness after treatment completion, with follow-up every 3-6 months for 2 years or until death.

2 years
Every 3-6 months

Treatment Details

Interventions

  • Darolutamide (Androgen Receptor Inhibitor)
  • Leuprolide Acetate (Gonadotropin-releasing Hormone Agonist)
Trial OverviewThe trial is testing darolutamide combined with leuprolide acetate in patients with salivary gland cancer driven by androgens. Darolutamide blocks the effects of androgens on cancer cells while leuprolide decreases hormone levels in the body. The goal is to see if this combination can stop tumor growth or shrink them.
Participant Groups
1Treatment groups
Experimental Treatment
Group I: Treatment (darolutamide, leuprolide acetate)Experimental Treatment6 Interventions
Patients receive darolutamide PO BID on days 1-28 of each cycle and leuprolide acetate IM every 4 or 12 weeks. Cycles repeat every 28 days in the absence of disease progression or unacceptable toxicity. Patients also undergo biopsy, collection of blood samples, and CT/MRI throughout the trial.

Darolutamide is already approved in Canada for the following indications:

🇨🇦
Approved in Canada as Nubeqa for:
  • Non-metastatic castration-resistant prostate cancer (nmCRPC)
  • Metastatic hormone-sensitive prostate cancer (mHSPC) in combination with docetaxel

Find a Clinic Near You

Research Locations NearbySelect from list below to view details:
University of Wisconsin Carbone Cancer Center - Eastpark Medical CenterMadison, WI
Los Angeles County-USC Medical CenterLos Angeles, CA
University of Colorado HospitalAurora, CO
University of Wisconsin Carbone Cancer Center - University HospitalMadison, WI
More Trial Locations
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Who Is Running the Clinical Trial?

National Cancer Institute (NCI)

Lead Sponsor

Trials
14080
Patients Recruited
41,180,000+

Findings from Research

Darolutamide: First Approval.Markham, A., Duggan, S.[2020]
In a 6-month study involving 117 patients with prostate cancer, the 3-month subcutaneous depot of leuprolide acetate (LA-2550) effectively suppressed serum testosterone levels to below 50 ng/dl in 98% of patients by day 28, and all patients achieved this level by day 35.
The treatment was well-tolerated, with no flare reactions and minimal adverse effects, primarily mild to moderate hot flashes, indicating a favorable safety profile while achieving significant reductions in testosterone and prostate-specific antigen levels.
A clinical study of 22.5 mg. La-2550: A new subcutaneous depot delivery system for leuprolide acetate for the treatment of prostate cancer.Chu, FM., Jayson, M., Dineen, MK., et al.[2023]
Darolutamide: A Review in Metastatic Hormone-Sensitive Prostate Cancer.Lee, A.[2023]
Darolutamide and Survival in Metastatic, Hormone-Sensitive Prostate Cancer.Smith, MR., Hussain, M., Saad, F., et al.[2023]
Darolutamide as a Second-Generation Androgen Receptor Inhibitor in the Treatment of Prostate Cancer.Abbasi, A., Movahedpour, A., Amiri, A., et al.[2021]
Darolutamide: A Review in Non-Metastatic Castration-Resistant Prostate Cancer.Scott, LJ.[2022]
Clinical Development of Darolutamide: A Novel Androgen Receptor Antagonist for the Treatment of Prostate Cancer.Fizazi, K., Smith, MR., Tombal, B.[2019]
In a phase 3 trial involving 1509 men with nonmetastatic, castration-resistant prostate cancer, darolutamide significantly improved median metastasis-free survival (40.4 months) compared to placebo (18.4 months).
At 3 years, overall survival was 83% in the darolutamide group versus 77% in the placebo group, with a 31% lower risk of death for those receiving darolutamide, while the incidence of adverse events was similar between both groups.
Nonmetastatic, Castration-Resistant Prostate Cancer and Survival with Darolutamide.Fizazi, K., Shore, N., Tammela, TL., et al.[2021]
Darolutamide in Nonmetastatic, Castration-Resistant Prostate Cancer.Fizazi, K., Shore, N., Tammela, TL., et al.[2022]

References

Darolutamide: First Approval. [2020]
A clinical study of 22.5 mg. La-2550: A new subcutaneous depot delivery system for leuprolide acetate for the treatment of prostate cancer. [2023]
Darolutamide: A Review in Metastatic Hormone-Sensitive Prostate Cancer. [2023]
Darolutamide and Survival in Metastatic, Hormone-Sensitive Prostate Cancer. [2023]
Darolutamide as a Second-Generation Androgen Receptor Inhibitor in the Treatment of Prostate Cancer. [2021]
Darolutamide: A Review in Non-Metastatic Castration-Resistant Prostate Cancer. [2022]
Clinical Development of Darolutamide: A Novel Androgen Receptor Antagonist for the Treatment of Prostate Cancer. [2019]
Nonmetastatic, Castration-Resistant Prostate Cancer and Survival with Darolutamide. [2021]
Darolutamide in Nonmetastatic, Castration-Resistant Prostate Cancer. [2022]